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all targets
· 60 indexed
Suggest a Target →
Suggest a Target
Target Name *
Alternative Names
UniProt ID
(optional)
Effect Type
(pick 1–3)
muscle
weight loss
pain
skin
diabetes
cancer
brain
cardiovascular
immune
gut
reproductive
aging
sleep
inflammation
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ALL
60
MUSCLE
10
WEIGHT LOSS
9
PAIN
4
SKIN
4
DIABETES
4
CANCER
4
BRAIN
7
CARDIOVASCULAR
4
IMMUNE
1
GUT
4
REPRODUCTIVE
4
AGING
12
SLEEP
2
INFLAMMATION
7
metalloprotease
ACE
angiotensin-converting enzyme
cardiovascular
cards
502
authors
1
cytoskeletal protein
Actin (G-actin)
G-actin
muscle
cards
2
authors
1
TGF-β superfamily
Activin A
INHBA
muscle · aging · inflammation
cards
3
authors
1
TGF-β superfamily
ActRIIB
activin receptor type 2B
muscle · aging
cards
2
authors
1
secretin-like GPCR (class B)
ADCYAP1R1 / PAC1R
PAC1 receptor
pain · brain · inflammation
cards
13
authors
1
CATEGORY
Anti-Aging
longevity
aging · skin
cards
1
authors
1
CATEGORY
Anticancer
cancer
cards
199
authors
1
CATEGORY
Antimicrobial
AMP
immune · inflammation
cards
301
authors
1
rhodopsin-like GPCR (class A)
AVPR2
vasopressin V2 receptor
cardiovascular
cards
7
authors
1
orphan-receptor ligand
BRP-R
weight loss · anti-obesity
cards
1
authors
1
secretin receptor family (class B GPCR)
CALCR/RAMP
calcitonin receptor
pain · cardiovascular
cards
31
authors
1
lipid target
Cardiolipin
inner mitochondrial membrane
aging
cards
2
authors
1
rhodopsin-like GPCR (class A)
CCKAR
CCK1 receptor
gut · weight loss
cards
26
authors
1
CATEGORY
Cosmeceutical
skin
cards
6
authors
1
secretin-like GPCR (class B)
CRHR2
CRF2 receptor
brain · weight loss
cards
16
authors
1
rhodopsin-like GPCR (class A)
EDNRA
ETA receptor
cardiovascular
cards
19
authors
1
type I cytokine receptor superfamily
EPOR
erythropoietin receptor
cardiovascular · inflammation
cards
2
authors
1
glycoprotein hormone receptor (class A GPCR)
FSHR
FSH receptor
sexual health
cards
1
authors
1
rhodopsin-like GPCR (class A)
GALR1
galanin-1 receptor
brain · gut · weight loss
cards
17
authors
1
secretin receptor family (class B GPCR)
GCGR
glucagon receptor
weight loss · diabetes
cards
23
authors
1
TGF-β superfamily
GDF-11
growth differentiation factor 11
muscle · aging
cards
2
authors
1
TGF-β superfamily
GDF-8
myostatin
muscle · weight loss · aging
cards
3
authors
1
best
0.742
Class B GPCR / secretin receptor family
GHRHR
cards
3
authors
1
endocrine
GH Secretagogue
GHRH
muscle · aging
cards
1
authors
1
rhodopsin-like GPCR (class A)
GHSR
ghrelin receptor
muscle · gut · sleep
cards
21
authors
1
secretin receptor family (class B GPCR)
GIPR
GIP receptor
weight loss · diabetes
cards
14
authors
1
secretin receptor family (class B GPCR)
GLP-1R
GLP-1 receptor
weight loss · diabetes · gut
cards
229
authors
1
secretin-like GPCR (class B)
GLP-2R
glucagon-like peptide 2 receptor
gut
cards
11
authors
1
rhodopsin-like (class A GPCR)
GnRHR
GnRH receptor
cancer · sexual health
cards
12
authors
1
rhodopsin-like GPCR (class A)
GPR173
SREB3
cards
1
authors
1
receptor tyrosine kinase
IGF-1R
insulin-like growth factor 1 receptor
muscle · cancer · aging
cards
7
authors
1
CATEGORY
Immune
cards
3
authors
1
receptor tyrosine kinase
INSR
insulin receptor
diabetes · aging
cards
3
authors
1
K2P (two-pore-domain) potassium channel family
KCNK2 / TREK-1
cards
1
authors
1
rhodopsin-like GPCR (class A)
KISS1R
kisspeptin receptor
sexual health · brain
cards
8
authors
1
glycoprotein hormone receptor (class A GPCR)
LHCGR
LH receptor
sexual health
cards
5
authors
1
CATEGORY
Longevity
aging
cards
7
authors
1
rhodopsin-like GPCR (class A)
MC1R
melanocortin-1 receptor
skin · inflammation
cards
5
authors
2
rhodopsin-like GPCR (class A)
MC2R
melanocortin-2 receptor
cardiovascular
cards
17
authors
1
rhodopsin-like GPCR (class A)
MC3R
melanocortin-3 receptor
weight loss · brain
cards
22
authors
1
rhodopsin-like GPCR (class A)
MC4R
melanocortin-4 receptor
weight loss · sexual health · brain
cards
18
authors
1
CATEGORY
Mitochondrial
MDP
muscle · aging
cards
1
authors
1
CATEGORY
Neuroprotective
nootropic
brain
cards
8
authors
1
rhodopsin-like GPCR (class A)
NPBWR1
neuropeptide B receptor 1
brain · pain
cards
13
authors
1
Class A GPCR / RFamide receptor family
NPFFR2
cards
1
authors
1
rhodopsin-like GPCR (class A)
NTSR1
neurotensin-1 receptor
brain · gut
cards
29
authors
1
rhodopsin-like GPCR (class A)
OPRD1
delta-opioid receptor
pain · brain
cards
18
authors
1
rhodopsin-like GPCR (class A)
OPRM1
mu-opioid receptor
pain
cards
33
authors
1
best
4
class A GPCR
OX2R
wakefulness · arousal · energy-homeostasis
cards
2
authors
1
rhodopsin-like GPCR (class A)
OXTR
oxytocin receptor
brain · sexual health
cards
4
authors
1
secretin-like GPCR (class B)
PTH1R
PTH receptor type 1
cardiovascular · aging
cards
25
authors
1
Class A GPCR / lysophospholipid receptor family
S1PR2
cards
1
authors
1
secretin-like GPCR (class B)
SCTR
secretin receptor
gut · brain
cards
6
authors
1
CATEGORY
Skin Peptides
cosmeceutical
skin
cards
3
authors
1
SSTR2
endocrine
cards
1
authors
1
rhodopsin-like GPCR (class A)
TACR1
NK1 receptor
pain · brain · inflammation
cards
19
authors
1
rhodopsin-like GPCR (class A)
TACR2
NK2 receptor
pain · gut · inflammation
cards
10
authors
1
CATEGORY
Tissue Repair
wound healing
inflammation · aging
cards
5
authors
1
rhodopsin-like GPCR (class A)
UTS2R
urotensin II receptor
cardiovascular
cards
1
authors
1
secretin receptor family (class B GPCR)
VPAC1
VIP receptor 1
brain · inflammation · gut
cards
26
authors
1